I-Albendazole iyi-anthelmintic yokwenziwa eseqenjini le-benzimidazole-derivatives elinomsebenzi olwa nezinhlobonhlobo zezikelemu kanye nezinga eliphakeme lokulinganisa futhi nasezigabeni zabantu abadala zesibindi.
I-Albendazole ihlangene neprotheni ye-eelworm's microtubule futhi ibambe iqhaza. Ngemuva kokuthi i-albenzene ihlanganiswe ne-β- tubulin, ingavimbela ukuncipha phakathi kwe-albenzene ne-α i-tubulin ehlangana ibe ama-microtubules. Ama-microtubules ayisakhiwo esiyisisekelo samayunithi amaningi amaseli. Ukusondelana kwe-Albendazole ne-nematodes tubulin kuphakeme kakhulu kunokuhlangana kwe-mammalian tubulin, ngakho-ke ubuthi kumammalia buncane.
I-Prophylaxis kanye nokwelashwa kwezifo ezinesifo emathunjini nasezinkomeni ezifana:
Izikelemu zesisu: I-Bunostomum, i-Cooperia, i-Chabertia, i-Haemonchus, i-Nematodirus, i-Oesophagostomum, i-Ostertagia, i-Strongyloides ne-Trichostrongylus spp.
Izibungu zamaphaphu: UDictyocaulus viviparus noD. Filaria.
Izikelemu zesikhunta: Monieza spp.
Isibindi-i-fluke: umuntu omdala uFasciola hepatica.
I-Albendazole nayo inomphumela we-ovicidal.
Ukuphatha ezinsukwini zokuqala ezingama-45 zokukhulelwa.
Ukusabela kwe-Hypersensitivity.
Ukuphathwa ngomlomo.
Okwezikelemu, izikelemu:
Izinkomo / izinyathi / ihhashi / izimvu / imbuzi: 5mg / kg bodyweight
Inja / ikati: 10 to 25mg / kg bodyweight
Okwezikhukhula:
Izinkomo / izinyathi: 10mg / kg bodyweight
Izimvu / imbuzi: 7.5mg / kg isisindo somzimba
Amathole nezinkomo: i-bolus eyodwa nge-300 kg. isisindo somzimba.
Okwesibindi-i-fluke:
1 bolus ngama-250 kg ngamunye. isisindo somzimba.
Gcina lapho izingane zingafinyeleli khona.
3 iminyaka.
- Okwenyama: Izinsuku eziyi-12.
- Okobisi: 4 izinsuku.
Gcina endaweni epholile, eyomile evikelwe ekukhanyeni.
Ikhwalithi yokuqala, Ukuphepha kuqinisekisiwe